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Found 139 Enz. Inhib. hit(s) with Target = 'Follicle-stimulating hormone receptor'
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410306(CHEMBL436481)
Affinity DataIC50:  5nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410307(CHEMBL360981)
Affinity DataIC50:  5nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410303(CHEMBL361847)
Affinity DataIC50:  7nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410309(CHEMBL365545)
Affinity DataIC50:  9nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50162936(Biphenyl-4-carboxylic acid (1-acetyl-2,2,4-trimeth...)
Affinity DataIC50:  10nMAssay Description:In vitro inhibition of maximum response evoked by cAMP on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50614128(CHEMBL5281228)
Affinity DataIC50:  17nMAssay Description:Allosteric antagonist activity at human FSHR expressed in CHO cells assessed as inhibition of FSH-induced activity incubated for 4 hrs by CRE-lucifer...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410304(CHEMBL195469)
Affinity DataIC50:  25nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410302(CHEMBL361167)
Affinity DataIC50:  27nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50162936(Biphenyl-4-carboxylic acid (1-acetyl-2,2,4-trimeth...)
Affinity DataIC50:  28nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50162936(Biphenyl-4-carboxylic acid (1-acetyl-2,2,4-trimeth...)
Affinity DataIC50:  28nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410308(CHEMBL192868)
Affinity DataIC50:  30nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410298(CHEMBL178980)
Affinity DataIC50:  31nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50335479((R)-N-(1-acetyl-2,2,4-trimethyl-4-(4-(prop-2-ynylo...)
Affinity DataIC50:  39nMAssay Description:Agonist activity at human FSHR receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410294(CHEMBL195347)
Affinity DataIC50:  50nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410292(CHEMBL192334)
Affinity DataIC50:  54nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50614109(CHEMBL5285685)
Affinity DataIC50:  64nMAssay Description:Antagonist activity at human FSHR expressed in HEK293 cells assessed as reduction in cAMP production incubated for 2 hrs by Eu-cAMP tracer based TR-F...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410300(CHEMBL179505)
Affinity DataIC50:  76nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50614127(CHEMBL5267043)
Affinity DataIC50:  156nMAssay Description:Antagonist activity at human FSHR expressed in HEK293 cells assessed as reduction in cAMP production incubated for 2 hrs by Eu-cAMP tracer based TR-F...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410297(CHEMBL372649)
Affinity DataIC50:  166nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410299(CHEMBL426824)
Affinity DataIC50:  170nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50614110(CHEMBL5270266)
Affinity DataIC50:  214nMAssay Description:Antagonist activity at human FSHR expressed in HEK293 cells assessed as reduction in cAMP production incubated for 2 hrs by Eu-cAMP tracer based TR-F...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410296(CHEMBL363164)
Affinity DataIC50:  240nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50614108(CHEMBL5290721)
Affinity DataIC50:  259nMAssay Description:Antagonist activity at human FSHR expressed in HEK293 cells assessed as reduction in cAMP production incubated for 2 hrs by Eu-cAMP tracer based TR-F...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50614104(CHEMBL5283477)
Affinity DataIC50:  270nMAssay Description:Antagonist activity at human FSHR expressed in HEK293 cells assessed as reduction in cAMP production incubated for 2 hrs by Eu-cAMP tracer based TR-F...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50614122(CHEMBL5273361)
Affinity DataIC50:  322nMAssay Description:Antagonist activity at human FSHR expressed in HEK293 cells assessed as reduction in cAMP production incubated for 2 hrs by Eu-cAMP tracer based TR-F...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50335480((R)-N-(1-acetyl-4-(4-((1-(2-(2-(2-azidoethoxy)etho...)
Affinity DataIC50:  324nMAssay Description:Agonist activity at human FSHR receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50614106(CHEMBL5275619)
Affinity DataIC50:  432nMAssay Description:Antagonist activity at human FSHR expressed in HEK293 cells assessed as reduction in cAMP production incubated for 2 hrs by Eu-cAMP tracer based TR-F...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50614105(CHEMBL5287707)
Affinity DataIC50:  449nMAssay Description:Antagonist activity at human FSHR expressed in HEK293 cells assessed as reduction in cAMP production incubated for 2 hrs by Eu-cAMP tracer based TR-F...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50614121(CHEMBL5280508)
Affinity DataIC50:  458nMAssay Description:Antagonist activity at human FSHR expressed in HEK293 cells assessed as reduction in cAMP production incubated for 2 hrs by Eu-cAMP tracer based TR-F...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50614111(CHEMBL5279687)
Affinity DataIC50:  466nMAssay Description:Antagonist activity at human FSHR expressed in HEK293 cells assessed as reduction in cAMP production incubated for 2 hrs by Eu-cAMP tracer based TR-F...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetFollicle-stimulating hormone receptor(Rattus norvegicus)
Research And Development

Curated by ChEMBL
LigandPNGBDBM50162936(Biphenyl-4-carboxylic acid (1-acetyl-2,2,4-trimeth...)
Affinity DataIC50:  540nMAssay Description:In vitro inhibition against maximum response evoked by cAMP in rat GFSHR-17 granulosa cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410301(CHEMBL372506)
Affinity DataIC50:  580nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50614113(CHEMBL5275140)
Affinity DataIC50:  606nMAssay Description:Antagonist activity at human FSHR expressed in HEK293 cells assessed as reduction in cAMP production incubated for 2 hrs by Eu-cAMP tracer based TR-F...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50614117(CHEMBL5275472)
Affinity DataIC50:  912nMAssay Description:Antagonist activity at human FSHR expressed in HEK293 cells assessed as reduction in cAMP production incubated for 2 hrs by Eu-cAMP tracer based TR-F...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50335470((R)-4-(3-(2-((1-(2-(2-(2-(4-((4-(1-acetyl-6-biphen...)
Affinity DataIC50:  920nMAssay Description:Agonist activity at human FSHR receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410291(CHEMBL194996)
Affinity DataIC50:  930nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50335472((R)-4-(3-(2-((1-(14-(4-((4-(1-acetyl-6-biphenyl-4-...)
Affinity DataIC50:  1.02E+3nMAssay Description:Agonist activity at human FSHR receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50614107(CHEMBL5288869)
Affinity DataIC50:  1.11E+3nMAssay Description:Antagonist activity at human FSHR expressed in HEK293 cells assessed as reduction in cAMP production incubated for 2 hrs by Eu-cAMP tracer based TR-F...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50614112(CHEMBL5267037)
Affinity DataIC50:  1.44E+3nMAssay Description:Antagonist activity at human FSHR expressed in HEK293 cells assessed as reduction in cAMP production incubated for 2 hrs by Eu-cAMP tracer based TR-F...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50335471((R)-4-(3-(2-((1-(2-(2-(2-(2-(4-((4-(1-acetyl-6-bip...)
Affinity DataIC50:  1.66E+3nMAssay Description:Agonist activity at human FSHR receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50614125(CHEMBL5270771)
Affinity DataIC50:  1.75E+3nMAssay Description:Antagonist activity at human FSHR expressed in HEK293 cells assessed as reduction in cAMP production incubated for 2 hrs by Eu-cAMP tracer based TR-F...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410293(CHEMBL195321)
Affinity DataIC50:  1.88E+3nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50614123(CHEMBL5286556)
Affinity DataIC50:  2.05E+3nMAssay Description:Antagonist activity at human FSHR expressed in HEK293 cells assessed as reduction in cAMP production incubated for 2 hrs by Eu-cAMP tracer based TR-F...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50614119(CHEMBL5271120)
Affinity DataIC50:  2.55E+3nMAssay Description:Antagonist activity at human FSHR expressed in HEK293 cells assessed as reduction in cAMP production incubated for 2 hrs by Eu-cAMP tracer based TR-F...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410295(CHEMBL371595)
Affinity DataIC50:  2.80E+3nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50614114(CHEMBL5268512)
Affinity DataIC50:  5.67E+3nMAssay Description:Antagonist activity at human FSHR expressed in HEK293 cells assessed as reduction in cAMP production incubated for 2 hrs by Eu-cAMP tracer based TR-F...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50614120(CHEMBL5267166)
Affinity DataIC50:  6.00E+3nMAssay Description:Antagonist activity at human FSHR expressed in HEK293 cells assessed as reduction in cAMP production incubated for 2 hrs by Eu-cAMP tracer based TR-F...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50559935(CHEMBL4780505)
Affinity DataIC50:  8.03E+3nMAssay Description:Antagonist activity at human FSHR expressed in CHO-K1 cells by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50614118(CHEMBL5288635)
Affinity DataIC50:  8.24E+3nMAssay Description:Antagonist activity at human FSHR expressed in HEK293 cells assessed as reduction in cAMP production incubated for 2 hrs by Eu-cAMP tracer based TR-F...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50614116(CHEMBL5285143)
Affinity DataIC50:  1.00E+4nMAssay Description:Antagonist activity at human FSHR expressed in HEK293 cells assessed as reduction in cAMP production incubated for 2 hrs by Eu-cAMP tracer based TR-F...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
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